- Used for the relief of dry, irritating, or unproductive cough, often associated with upper respiratory tract infections, bronchitis, or post-infectious cough. Provides antitussive, bronchodilatory, mucolytic, and antihistaminic effects.
- Dose:
- Adults: PO 5–10 mL every 6–8 hours
- Children 6–12 years: PO 2.5–5 mL every 6–8 hours
- Children <6 years: Not recommended due to risk of respiratory depression from codeine and promethazine
Suspension
- Codeine phosphate: 10 mg
- Ephedrine HCl: 15 mg
- Potassium guaiacolsulfonate: 100 mg
- Promethazine HCl: 5 mg
- Shake well before use
- Use a proper measuring device (not a kitchen spoon)
- Do not exceed 4 doses/day
- Avoid alcohol and other sedatives
- Stay hydrated to assist mucus clearance
- Codeine: Centrally acting opioid antitussive; suppresses cough reflex in the brain stem.
- Ephedrine: Sympathomimetic bronchodilator and nasal decongestant; stimulates β and α receptors.
- Potassium Guaiacolsulfonate: An expectorant; helps liquefy mucus, facilitating its expulsion.
- Promethazine: First-generation antihistamine with strong sedative, anticholinergic, and antiemetic effects.
- Codeine: Drowsiness, constipation, nausea, dizziness, respiratory depression (especially in overdose or ultra-rapid metabolizers)
- Ephedrine: Hypertension, tachycardia, insomnia, tremors, anxiety
- Hypersensitivity to any component
- Children <12 years (codeine risk of severe respiratory events)
- Respiratory depression, bronchial asthma in acute attack
- MAO inhibitor use within 14 days (ephedrine interaction)
- Prostatic hypertrophy, bladder neck obstruction, or glaucoma (promethazine caution)
- Severe hepatic impairment (due to codeine metabolism)
- MAO inhibitors: Risk of hypertensive crisis (ephedrine)
- Other CNS depressants (benzodiazepines, alcohol): Additive sedation and respiratory depression
- CYP2D6 inhibitors: May alter codeine metabolism
Anticholinergic drugs: Additive effects with promethazine
Drug Status
Availability | prescription, controlled,scheduled |
Pregnancy | Not recommended unless absolutely necessary |
Breastfeeding | Avoid during breastfeeding |
Schedule | yes |
BRAND NAME | STRENGTH | FORMULATION | PACK SIZE | MANUFACTURER | DISTRIBUTOR |
---|---|---|---|---|---|
Codelzine Linctus | 8mg/8mg/25mg/4mg per 5mL | Suspension | 60mL, 100mL | Elys Chemicals | Elys Chemicals |