• Chronic angina:
    • Initially PO 500mg BD
    • Max: 2000mg/day
  • Tablet:
    • 375mg
    • 500mg
    • 750mg
    • 1000mg

Taken without regards to meals

Non-nitrate antianginal

It is thought to inhibit late sodium current, reducing sodium-induced calcium overload in myocytes

  • Dizziness
  • Headache
  • Constipation
  • Nausea
  • Asthenia
  • Palpitations
  • Tinnitus
  • Vertigo
  • Blurred vision
  • Abdominal pain
  • Xerostomia
  • Vomiting
  • Dyspepsia
  • Peripheral edema
  • Anorexia
  • Confusion
  • Dyspnea
  • Hyperhidrosis
  • Hypersensitivity to components
  • Cirrhosis
  • Apalutamide
  • Atazanavir
  • Bosentan
  • Butabarbital
  • Butalbital
  • Carbamazepine
  • Cenobamate
  • Ceritinib
  • Chloramphenicol
  • Cisapride
  • Clarithromycin
  • Cobicistat
  • Dabrafenib
  • Darunavir
  • Dofetilide
  • Efavirenz
  • Enzalutamide
  • Etravirine
  • Fosphenytoin
  • Idelalisib
  • Itraconazole
  • Ketoconazole
  • Levoketoconazole
  • Lonafarnib
  • Lopinavir/ritonavir
  • Lorlatinib
  • Lumacaftor/ivacaftor
  • Mavacamten
  • Mifepristone
  • Mitapivat
  • Mitotane
  • Modafinil
  • Nafcillin
  • Nefazodone
  • Nelfinavir
  • Pentobarbital
  • Pexidartinib
  • Phenobarbital
  • Phenytoin
  • Pimozide
  • Posaconazole
  • Primidone
  • Ribociclib
  • Rifabutin
  • Rifampin
  • Rifapentine
  • Ritonavir
  • Saquinavir
  • Sotorasib
  • Thioridazine
  • Tipranavir
  • Tucatinib
  • Voriconazole

                          Drug Status

Availability Prescription only
Pregnancy Category C; Weigh risk vs benefits
Breastfeeding Contraindicated
Schedule Not controlled
BRAND NAME STRENGTH FORMULATION PACK SIZE MANUFACTURER DISTRIBUTOR
Cartinex-OD 1g Tablet 30’s Micro Labs India Micro Labs
Ranexa 375mg Tablet 60’s Menarini International Phillips Therapeutics
Ranexa 500mg Tablet 60’s Menarini International Phillips Therapeutics
Ranexa 750mg Tablet 60’s Menarini International Phillips Therapeutics