- Invasive intestinal amebiasis:
- Adults: PO 800mg TDS *5-10 days
- 7-10 yrs: PO 400mg TDS * 5/7
- 3-7 yrs: 200mg QID *5/7
- 1-3yrs: 200mg TDS*5/7
- Eradication of cysts in symptomless carriers:
- PO 400mg-800mg TDS *5-10 days
- Prophylaxis of post-operative infections:
- Adults & >12 yrs: PO 1g TDS day prior to surgery OR IV 500mg*1, 60 min prior to surgery
- <12yrs: PO 20-30mg/kg (maximum 500mg) single dose, 1-2 hrs before surgery
- Treatment of urogenital trichomoniasis:
- Adults & >10 yrs: PO 200mg TDS *1/52 OR PO 400mg BD *5-7 days OR PO 2g as a single dose.
- Sexual partners should receive similar concurrent treatment
- 7 -10 yrs: PO 100mg TDs*1/52
- 3-7 yrs: PO 100mg BD *1/52
- 1-3 yrs: PO 50mg TDS *1/52
- Adults & >10 yrs: PO 200mg TDS *1/52 OR PO 400mg BD *5-7 days OR PO 2g as a single dose.
- Bacterial vaginosis:
- PO 400mg BD *5-7 days OR PO 2g*1
- Pelvic Inflammatory Disease:
- PO 400mg BD OR IV 500mg BD *14/7
- Bacterial vaginosis:
- PO 400mg BD *1/52 OR 2g *1
- PO 250mg TDS *1/52 in pregnant patients
- Giardiasis:
- Adults: PO 2g OD *3/7 OR PO 400mg TDS *5/7
- 7-10 yrs: PO 1g *3/7
- 3-7 yrs: PO 600-800mg OD *3/7
- 1-3 yrs: PO 500mg OD *3/7
- Acute ulcerative gingivitis/ dental infections:
- Adults: PO 400mg TDS *3/7
- 10-18 yrs: PO 200mg-250mg TDS * 3-7 days.
- 7-10 yrs: PO 100mg TDS * 3-7 days.
- 3-7 yrs: PO 100mg BD * 3-7 days
- 1-3 yrs: PO 50mg TDS * 3-7 days.
- Leg ulcers/pressure sores:
- Adults: PO 400mg TDS *1/52
- 12 -18 yrs: PO 400mg BD* 14/7
- Amebiasis:
- Adults: PO 800mg TDS*5/7
- 7-10yrs: PO 400mg TDS*5/7
- 3-7 yrs: PO 200mg QID *5/7
- 1-3 yrs: PO 200mg TDS*5/7
- Tablet:
- 200mg
- 400mg
- Suspension:
- 200mg/5mL
- Injection:
- 0.5% w/v
- Avoid alcohol while taking medication and for at least three days after discontinuation.
- To prevent stomach upset, take this medication with food or a full glass of water or milk.
Nitroimidazole
It acts by inhibiting nucleic acid synthesis by disrupting DNA and causing strand breakage; amoebicidal, bactericidal and trichomonacidal. Active against: Balantidium coli, Blastocystis hominis, Entamoeba histolytica, Giardia lambia and Trichomonas vaginalis. Also active against Bacteroides and Clostridium spp.
- GI disturbances especially nausea
- Metallic taste
- Headache
- Anorexia
- Vomiting
- Diarrhea
- Dry mouth
- Furred tongue
- Darkened urine
- Transient fall in BP
- Bone marrow depression
- Vertigo
- Dizziness
- Depression
- Insomnia.
- Pseudomembranous colitis
- Hypersensitive reactions
- Concurrent antihypertensive therapy
- Alcohol
- Disulfiram
- Lopinavir/ritonavir
- Lithium
Drug Status
Availability | Prescription or OTC by Pharmacist |
Pregnancy | Category B2; Contraindicated |
Breastfeeding | Contraindicated |
Schedule | Not controlled |
BRAND NAME | STRENGTH | FORMULATION | PACK SIZE | MANUFACTURER | DISTRIBUTOR |
---|---|---|---|---|---|
Abagyl | 0.5% w/v | Injection | 100mL | Abacus Pharma | Abacus Pharma |
Amebazole | 200mg/5mL | Suspension | 60mL, 100mL | Sphinx Pharma | Sphinx Pharma |
Amebazole | 400mg | Tablet | 100’s | Sphinx Pharma | Sphinx Pharma |
Amebazole | 200mg | Tablet | 250’s | Sphinx Pharma | Sphinx Pharma |
Amebil | 200mg/5mL | Suspension | 60mL, 100mL | Njimia Ltd | Njimia Ltd |
Amizole | 200mg/5mL | Suspension | 60mL, 100mL | Biopharma Ltd | Biopharma Ltd |
Amizole | 200mg | Tablet | 100’s, 1000’s | Biopharma Ltd | Biopharma Ltd |
Amizole | 400mg | Tablet | 100’s | Biopharma Ltd | Biopharma Ltd |
Axagyl | 0.5% w/v | Injection | 100mL | Axa Parenterals | Axa Parenterals |
Dangyl | 200mg | Tablet | 100’s | Dinlas Pharma | Dinlas Pharma |
Dangyl | 200mg/5mL | Suspension | 60mL, 100mL | Dinlas Pharma | Dinlas Pharma |
Eflaron | 400mg | Tablet | 100’s | Dawa Ltd | Dawa Ltd |
Eflaron | 200mg/5mL | Suspension | 60mL, 100mL | Dawa Ltd | Dawa Ltd |
Eflaron | 200mg | Tablet | 100’s | Dawa Ltd | Dawa Ltd |
Elogyl | 200mg | Tablet | 100’s | Elys Chemicals | Elys Chemicals |
Elogyl | 400mg | Tablet | 100’s | Elys Chemicals | Elys Chemicals |
Elogyl | 200mg/5mL | Suspension | 60mL, 100mL | Elys Chemicals | Elys Chemicals |
Filmet | 200mg/5mL | Suspension | 60mL | Beximco Pharma | Madawa Pharma |
Flagimed | 200mg/5mL | Suspension | 60mL, 100mL | Medivet Products | Medivet Products |
Flagyl | 200mg/5mL | Suspension | 100mL | Sanofi-Aventis | Ressourcethica Kenya |
Flagyl | 400mg | Tablet | 100’s | Sanofi-Aventis | Ressourcethica Kenya |
Flagyl | 0.5% w/v | Injection | 100mL | Sanofi-Aventis | Ressourcethica Kenya |
Medzol | 400mg | Tablet | 100’s, 400’s | Careplus Ltd | Careplus Ltd |
Megyl | 400mg | Tablet | 100’s | Regal Pharma | Regal Pharma |
Megyl | 200mg | Tablet | 100’s | Regal Pharma | Regal Pharma |
Megyl | 200mg per 5mL | Suspension | 100mL | Regal Pharma | Regal Pharma |
Metris | 0.5% w/v | Injection | 100mL | Claris Otsuka | Reddys Pharma |
Metris | 0.5% w/v | Injection | 100mL | Claris Otsuka | Reddys Pharma |
Metrogyl | 200mg | Tablet | 100’s | Unique Pharma | Harley’s Ltd |
Metrogyl | 0.5% w/v | Injection | 100mL | Unique Pharma | Harley’s Ltd |
Metronidazole | 0.5% w/v | Injection | 100mL | Abaris Healthcare | Unisel Ltd |
Metronidazole | 0.5% w/v | Injection | 100mL | Tasa Pharma | Tasa Pharma |
Metronidazole | 0.5% w/v | Injection | 100mL | Amanta Healthcare C/O Surgilinks | Surgilinks Ltd |
Metrowin | 200mg | Tablet | 1000’s | Medisel Kenya | Medisel Kenya |
Metrozol | 400mg | Tablet | 100’s | Cosmos Ltd | Cosmos Ltd |
Metrozol | 400mg | Tablet | 100’s | Cosmos Ltd | Cosmos Ltd |
Metzole | 0.5% w/v | Injection | 100mL | Global Pharma | Medox Pharma |
Mindazole | 0.5% w/v | Injection | 100mL | Kilitch Drugs | Nedah Pharma |
Nelzole | 200mg/5mL | Suspension | 60mL | Universal Corporation | Universal Corporation |
Nirmet | 0.5% w/v | Injection | 100mL | Aculife Healthcare | Crown Healthcare |
Shelgyl-200 | 200mg | Tablet | 1000’s | Shelys Pharma | Beta Healthcare |
Trichazole | 0.5% w/v | Injection | 100mL | Fresenius Kabi | Surgipharm Ltd |
Trichogyl | 0.5% w/v | Injection | 100mL | Til Healthcare | Harley’s Ltd |
Tricozole | 200mg | Tablet | 100’s | Laboratory & Allied | Laboratory & Allied |
Tricozole | 400mg | Tablet | 100’s | Laboratory & Allied | Laboratory & Allied |
Tricozole | 200mg/5mL | Suspension | 60mL, 100mL | Laboratory & Allied | Laboratory & Allied |
Trogyl | 200mg | Tablet | 100’s | Biodeal Labs | Biodeal Labs |
Trogyl | 400mg | Tablet | 100’s | Biodeal Labs | Biodeal Labs |
Trogyl | 200mg/5mL | Suspension | 60mL, 100mL | Biodeal Labs | Biodeal Labs |
Troz | 0.5% w/v | Injection | 100mL | Zawadi Healthcare | Zawadi Healthcare |