• Attention deficit hyperacidity disorder (ADHD):
    • PO 18-36mg OD OR 20-30mg/day divided BD/TDS
    • May increase by 18-mg increments at weekly intervals
    • Maintenance: 18-72mg/day
  • Narcolepsy:
    • PO 20-30mg/day divided BD/TDS
  • Tablet:
    • 10mg
    • 18mg
    • 27mg
    • 36mg
    • 54mg
  • Taken 30-45 minutes before meals

Norepinephrine-Dopamine Reuptake Inhibitors (NDRIs)

It stimulates CNS activity, blocks reuptake and increases release of norepinephrine and dopamine in extraneuronal space

  • Nervousness
  • Insomnia
  • Anorexia
  • Abdominal pain
  • Tachycardia
  • Nausea
  • Headache
  • Palpitations
  • Dizziness
  • Xerostomia
  • Irritability
  • Hyperhidrosis
  • Changes in BP
  • Changes in HR
  • Visual disturbance
  • Weight loss (long-term use)
  • Hypersensitivity to components/class
  • MAO inhibitor use within 14 days
  • Severe agitation
  • Severe anxiety
  • Motor tics
  • Tourette syndrome or family history
  • Severe cardiovascular disease
  • Cardiac structural abnormality
  • Severe arrhythmia
  • Cardiomyopathy
  • CAD
  • Glaucoma

WARNING:

  • Risk of abuse and dependence
  • Benzphetamine
  • Diethylpropion
  • Isocarboxazid
  • Linezolid
  • Phendimetrazine
  • Phenelzine
  • Phentermine
  • Rasagiline
  • Safinamide
  • Selegiline
  • Tranylcypromine

                          Drug Status

Availability Prescription only
Pregnancy Category D
Breastfeeding Weigh risk vs benefit
Schedule Controlled
BRAND NAME STRENGTH FORMULATION PACK SIZE MANUFACTURER DISTRIBUTOR
Concerta 18mg Tablet 30’s Janssen Pharmaceutica Janssen Pharmaceutica
Concerta 36mg Tablet 30’s Janssen Pharmaceutica Janssen Pharmaceutica
Concerta 27mg Tablet 30’s Janssen Pharmaceutica Janssen Pharmaceutica
Concerta 54mg Tablet 30’s Janssen Pharmaceutica Janssen Pharmaceutica
Ritalin 10mg Tablet 30’s Novartis Pharma Novartis Kenya