- Breast cancer:
- Node-positive adjuvant treatment:
- IV 75mg/m² 1 hour after doxorubicin and cyclophosphamide every 3 weeks x 6 cycles
- IV 75mg/m² 1 hour after doxorubicin and cyclophosphamide every 3 weeks x 6 cycles
- Node-positive adjuvant treatment:
-
- Monotherapy in locally advanced or metastatic cancer:
- IV 60-100mg/m² over 1 hour every 3 weeks
- IV 60-100mg/m² over 1 hour every 3 weeks
- Monotherapy in locally advanced or metastatic cancer:
-
- Metastatic disease, combined with capecitabine:
- IV 75mg/m²/dose**1 every 3 weeks
- For anthracycline-resistant disease
- Metastatic disease, combined with capecitabine:
- Locally advanced or metastatic non-small cell lung cancer:
- IV 75mg/m2 over 1 hour every 3 weeks
- IV 75mg/m2 over 1 hour every 3 weeks
- Hormone-refractory metastatic prostate cancer(castration resistant) in combination with prednisone:
- IV 75mg/m2 over 1 hour every 3 weeks with daily prednisone PO 5mg BD
- Up to 10 cycles
- Advanced gastric cancer in patients who have not received prior chemotherapy for advanced disease:
- Day 1: 75mg/m2 IV infusion over 1 hour then cisplatin 75mg/m2 as a 1-3 hr infusion
- Post cisplatin: Fluorouracil 750mg/m2 OD given as a 24-hr continuous infusion *5/7
- Repeat every 3 weeks
- Locally advanced squamous cell head/neck carcinoma:
- Day 1: 75mg/m2 IV infusion over 1 hour then cisplatin 75-100mg/m2 as a 1-3 hr infusion
- Post cisplatin: Fluorouracil 750mg/m2 OD given as a 24-hr continuous infusion *5/7
- Repeat every 3 weeks for 3-4 cycles
Injection:
- 20mg/mL
- 20mg/0.5mL
- 80mg/2mL
- 120mg/3mL
- To be used within 4 hours of dilution
- Non-PVC tubing used
- When administered as sequential infusions, taxane derivatives should be administered before platinum derivatives (cisplatin, carboplatin) to decrease risk of myelosuppression and to enhance efficacy
- Pre-medicate with dexamethasone
Taxane anticancer
It promotes formation and inhibits disassembly of stable microtubules thereby inhibiting mitosis
- Neutropenia
- Leukopenia
- Anemia
- Alopecia
- Asthenia
- Fluid retention
- Fatigue
- Nausea
- Diarrhea
- Sensory neuropathy
- Infection
- Nail changes
- Stomatitis
- Pharyngitis
- Taste changes
- Hyperbilirubinemia
- Elevated ALT/AST
- Vomiting
- Anorexia
- Dyspnea
- Arthralgia
- Myalgia
- Cough
- Lacrimation
- Rash
- Desquamation
- Hypersensitivity reaction
- Thrombocytopenia
- Constipation
- Pain
- Amenorrhea
- Hypersensitivity to class/components
- Hypersensitivity to polysorbate 80
- 1st trimester pregnancy
- Avoid breastfeeding during treatment and for 1 week after discontinuing
- ANC <1500
- Platelet count <100,000
- Bilirubin elevated
- ALT or AST >1.5x ULN with alk phos >2.5x ULN
WARNING:
- Increased mortality reported in patients with liver impairment
- Severe neutropenia with infection may occur
- Severe hypersensitivity reaction
- Severe fluid retention
- Use effective contraception during treatment and for 6 months after discontinuing in female patients and during treatment and for 3 months after discontinuing in male patients
- Live vaccines
- Disulfiram
- Metronidazole
- Topiramate
- Talimogene
Drug Status
Availability | Prescription only |
Pregnancy | Category D |
Breastfeeding | Contraindicated |
Schedule | Not controlled |
BRAND NAME | STRENGTH | FORMULATION | PACK SIZE | MANUFACTURER | DISTRIBUTOR |
---|---|---|---|---|---|
Adoxi | 20mg/0.5mL | Injection | 1’s | M/S Beta Drugs | Galaxy Pharma |
Adoxi | 80mg/2mL | Injection | 1’s | M/S Beta Drugs | Galaxy Pharma |
Adoxi | 120mg/3mL | Injection | 1’s | M/S Beta Drugs | Galaxy Pharma |
Celtere | 120mg/3mL | Injection | 1’s | Celon Labs | Europa Healthcare |
D-tail | 80mg | Injection | 1’s | PSM Pharma | PSM Pharma |
D-tail | 120mg | Injection | 1’s | PSM Pharma | PSM Pharma |
Docecord | 20mg/mL | Injection | 4mL | Intas Pharma | Accord Healthcare |
Docetax | 80mg/2mL | Injection | 1’s | Cipla Ltd | Imperial Managed |
Docetax | 20mg/0.5mL | Injection | 1’s | Cipla Ltd | Imperial Managed |
Docetec | 80mg/2mL | Injection | 1’s | United Biotech | Salama Pharma |
Docetec | 20mg/0.5mL | Injection | 1’s | United Biotech | Salama Pharma |
Doxol | 20mg/0.5mL | Injection | 1’s | Venus Remedies | Surgipharm Ltd |
Doxol | 80mg/2mL | Injection | 1’s | Venus Remedies | Surgipharm Ltd |
Doxol | 120mg/3mL | Injection | 1’s | Venus Remedies | Surgipharm Ltd |
Taceedo | 20mg/0.5mL | Injection | 1’s | Miracalus | Ripple Pharma |
Taceedo | 80mg/2mL | Injection | 1’s | Miracalus | Ripple Pharma |
Taceedo | 120mg/3mL | Injection | 1’s | Miracalus | Ripple Pharma |
Taxotere | 20mg/2mL | Injection | 1’s | Sanofi-Aventis | Ressourcethica Kenya |
Taxotere | 80mg/4mL | Injection | 1’s | Sanofi-Aventis | Ressourcethica Kenya |
Taxuba | 80mg/2mL | Injection | 1’s | Glenmark Pharma | Glenmark Pharma |
Taxuba | 20mg/0.5mL | Injection | 1’s | Glenmark Pharma | Glenmark Pharma |
Taxwell | 20mg/0.5mL | Injection | 1’s | Getwell Pharma | Nairobi Enterprises |
Taxwell | 80mg/2mL | Injection | 1’s | Getwell Pharma | Nairobi Enterprises |
Taxwell | 160mg/4mL | Injection | 1’s | Getwell Pharma | Nairobi Enterprises |